Drug Discovery

A novel combined experimental therapy in an Alzheimer's transgenic model
Investigator(s): A. Claudio Cuello, MD, DSc, FRSC
Institution(s): McGill University, Dept. of Pharmacology and Therapeutics
Duration: 2008 - 2009

Summary:

A number of strategies have been designed to lower the levels of amyloid beta in Alzheimer's disease (AD), in particular in the form of oligomers (molecular repeats of the Aβ amyloid protein. The investigator's laboratory has been able to repeat earlier work that reported partial clearance of Aβ in a transgenic model of AD using a compound called scyllo-inositol. In addition, the PI's laboratory has also revealed that the normal function of the neuroprotective nerve growth factor (NGF) is perturbed in transgenic models of AD and in AD human brain samples. This new finding may explain the selective vulnerability of NGF-dependent neurons involved in learning and memory to AD pathology. Preliminary data indicate that this dysfunction can be
controlled pharmacologically in animal models of AD. The PI's group have found remarkable beneficial effects of treating this novel target in conjunction with strategies to remove Aβ oligomers. The objective of this research proposal is to explore a novel combined therapy attacking simultaneously these two targets.

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